CGP71683 hydrochloride

CGP71683 hydrochloride (CGP71683A) is a competitive and sellective neuropeptide Y receptor type 5 (Y5 receptor) antagonist with Ki of 1.3 nM.

Product information

CAS Number: 192322-50-2

Molecular Weight: 512.07

Formula: C26H30ClN5O2S

Chemical Name: N-(((1r,4r)-4-(((4-aminoquinazolin-2-yl)amino)methyl)cyclohexyl)methyl)naphthalene-1-sulfonamide hydrochloride

Smiles: Cl.NC1=NC(NC[C@@H]2CC[C@@H](CNS(=O)(=O)C3=CC=CC4=CC=CC=C43)CC2)=NC2=CC=CC=C21

InChiKey: DIQDKUNCSVFGHH-VPLSKCCHSA-N

InChi: InChI=1S/C26H29N5O2S.ClH/c27-25-22-9-3-4-10-23(22)30-26(31-25)28-16-18-12-14-19(15-13-18)17-29-34(32,33)24-11-5-7-20-6-1-2-8-21(20)24;/h1-11,18-19,29H,12-17H2,(H3,27,28,30,31);1H/t18-,19-;

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Solubility: DMSO: 100 mg/mL(195.28 mM).

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 ^oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥12 months if stored properly.

Stock Solution Storage: 0 - 4 ^oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

References:

1. Anne Lecklin, et al. Br J Pharmacol. 2002 Apr;135(8):2029-37.

Products are for research use only. Not for human use.