CaMKII-IN-1

CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM; significantly high selectivity against CaMKIV, MLCK, p38a, Akt1, and PKC.

Product information

CAS Number: 1208123-85-6

Molecular Weight: 548.10

Formula: C29H30ClN5O2S

Chemical Name: N-{6-benzyl-2-[(2-phenylethyl)amino]-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl}-3-chloro-2-methylbenzene-1-sulfonamide

Smiles: CC1=C(Cl)C=CC=C1S(=O)(=O)NC1=NC(NCCC2C=CC=CC=2)=NC2CCN(CC3C=CC=CC=3)CC=21

InChiKey: LGUUETDTMQTHML-UHFFFAOYSA-N

InChi: InChI=1S/C29H30ClN5O2S/c1-21-25(30)13-8-14-27(21)38(36,37)34-28-24-20-35(19-23-11-6-3-7-12-23)18-16-26(24)32-29(33-28)31-17-15-22-9-4-2-5-10-22/h2-14H,15-20H2,1H3,(H2,31,32,33,34)

Technical Data

Appearance: Solid Power

Purity: ≥98% (or refer to the Certificate of Analysis)

Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis

Storage Condition: Dry, dark and -20 ^oC for 1 year or refer to the Certificate of Analysis.

Shelf Life: ≥360 days if stored properly.

Stock Solution Storage: 0 - 4 ^oC for 1 month or refer to the Certificate of Analysis.

Drug Formulation: To be determined

HS Tariff Code: 382200

Products are for research use only. Not for human use.