详情描述
CP-809101 is a potent and selective 5-HT2C receptor agonist (pEC50 values are 9.96, 7.19 and 6.81 for human 5-HT2C, 5-HT2B and 5-HT2A receptors respectively). CP-809101 reduce motor impulsivity and reinstatement of food seeking behavior in male rats. CP-809101 (0.3-3 mg/kg SC) reduced responding for both nicotine and food and blocked the discriminative stimulus properties of nicotine in a similar manner to lorcaserin and Ro 60-0175.
Product information
CAS Number: 1215721-40-6
Molecular Weight: 341.24
Formula: C15H18Cl2N4O
Chemical Name: 2-[(3-chlorophenyl)methoxy]-6-(piperazin-1-yl)pyrazine hydrochloride
Smiles: Cl.ClC1=CC(COC2=CN=CC(=N2)N2CCNCC2)=CC=C1
InChiKey: NMUNRTCTDLORDR-UHFFFAOYSA-N
InChi: InChI=1S/C15H17ClN4O.ClH/c16-13-3-1-2-12(8-13)11-21-15-10-18-9-14(19-15)20-6-4-17-5-7-20;/h1-3,8-10,17H,4-7,11H2;1H
Technical Data
Appearance: Solid Power
Purity: ≥98% (or refer to the Certificate of Analysis)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life: ≥360 days if stored properly.
Stock Solution Storage: 0 - 4 oC for 1 month or refer to the Certificate of Analysis.
Drug Formulation: To be determined
HS Tariff Code: 382200
Products are for research use only. Not for human use.